Publications | Drug Discovery Unit

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May 2019

Identification of inhibitors of an unconventional Trypanosoma brucei kinetochore kinase

Publication Date:
31 May 2019

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Characterising Covalent Warhead Reactivity. James S.Martin, Claire J.MacKenzie, Daniel Fletcher, Ian H.Gilbert

Publication Date:
15 May 2019

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A preclinical candidate for the treatment of visceral leishmaniasis that acts through proteasome inhibition. Wyllie et al.

Publication Date:
07 May 2019

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Optimisation of a Key Cross-Coupling Reaction Towards the Synthesis of a Promising Antileishmanial Compound

Publication Date:
02 May 2019

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Apr 2019

Lysyl-tRNA synthetase as a drug target in malaria and cryptosporidiosis

Publication Date:
02 Apr 2019

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Mar 2019

Discovery of Soft-Drug Topical Tool Modulators of Sphingosine-1-phosphate Receptor 1 (S1PR1)

Publication Date:
14 Mar 2019

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Feb 2019

A Continuous Flow Strategy for the Facile Synthesis and Elaboration of Semi-Saturated Heterobicyclic Fragments Nicola Luise, Eleanor W. Wyatt, Gary Tarver, Paul Wyatt

Publication Date:
14 Feb 2019

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Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis

Publication Date:
14 Feb 2019

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Jan 2019

Pharmacological validation of N-myristoyltransferase as a drug target in Leishmania donovani

Publication Date:
11 Jan 2019

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Dec 2018

Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis.

Publication Date:
20 Dec 2018

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Nov 2018

Pharmacological Validation of N-Myristoyltransferase as a Drug Target in Leishmania donovani.

Publication Date:
12 Nov 2018

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Oct 2018

Discovery of super soft-drug modulators of sphingosine-1-phosphate receptor 1.

Publication Date:
15 Oct 2018

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2,4-Diamino-6-methylpyrimidines for the potential treatment of Chagas’ disease.

Publication Date:
01 Oct 2018

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Sep 2018

Development of Chemical Proteomics for the Folateome and Analysis of the Kinetoplastid Folateome

Publication Date:
28 Sep 2018

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A Molecular Hybridization Approach for the Design of Potent, Highly Selective, and Brain-Penetrant N-Myristoyltransferase Inhibitors

Publication Date:
12 Sep 2018

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