Publications | Drug Discovery Unit

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Jul 2016

Molecular basis of RNA guanine-7 methyltransferase (RNMT) activation by RAM

Publication Date:
15 Jul 2016

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Identification of Novel Inhibitors of the Type I Interferon Induction Pathway Using Cell-Based High-Throughput Screening

Publication Date:
04 Jul 2016

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Jun 2016

Trisubstituted Pyrimidines as Efficacious and Fast-Acting Antimalarials

Publication Date:
27 Jun 2016

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Drug resistance in eukaryotic microorganisms

Publication Date:
24 Jun 2016

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Prediction of drug penetration in tuberculosis lesions

Publication Date:
22 Jun 2016

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May 2016

The anti-tubercular drug delamanid as a potential oral treatment for visceral leishmaniasis

Publication Date:
24 May 2016

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Apr 2016

Validation of N-myristoyltransferase as Potential Chemotherapeutic Target in Mammal-Dwelling Stages of Trypanosoma cruzi

Publication Date:
29 Apr 2016

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Identification of Trypanocidal Activity for Known Clinical Compounds Using a New Trypanosoma cruzi Hit-Discovery Screening Cascade

Publication Date:
15 Apr 2016

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Jan 2016

A Substrate Mimic Allows High-Throughput Assay of the FabA Protein and Consequently the Identification of a Novel Inhibitor of Pseudomonas aeruginosa FabA

Publication Date:
19 Jan 2016

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Nov 2015

A substrate mimic allows high throughput assay of the FabA protein and consequently the identification of a novel inhibitor of Pseudomonas aeruginosa FabA

Publication Date:
10 Nov 2015

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Oct 2015

Discovery of Indoline-2-carboxamide Derivatives as a New Class of Brain-Penetrant Inhibitors of Trypanosoma brucei

Publication Date:
05 Oct 2015

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Sep 2015

Development of Small-Molecule Trypanosoma brucei N-Myristoyltransferase Inhibitors: Discovery and Optimisation of a Novel Binding Mode

Publication Date:
28 Sep 2015

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Development and Validation of a Novel Leishmania donovani Screening Cascade for High-Throughput Screening Using a Novel Axenic Assay with High Predictivity of Leishmanicidal Intracellular Activity

Publication Date:
25 Sep 2015

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Development of a Fluorescence-based Trypanosoma cruzi CYP51 Inhibition Assay for Effective Compound Triaging in Drug Discovery Programmes for Chagas Disease.

Publication Date:
23 Sep 2015

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Discovery of Inhibitors of Trypanosoma brucei by Phenotypic Screening of a Focused Protein Kinase Library

Publication Date:
22 Sep 2015

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