Publications | Drug Discovery Unit

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Sep 2015

Discovery of Inhibitors of Trypanosoma brucei by Phenotypic Screening of a Focused Protein Kinase Library

Publication Date:
22 Sep 2015

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Jun 2015

A novel multiple-stage antimalarial agent that inhibits protein synthesis

Publication Date:
18 Jun 2015

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Apr 2015

Identification and structure solution of fragment hits against kinetoplastid N-myristoyltransferase.

Publication Date:
21 Apr 2015

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Feb 2015

N-Myristoyltransferase Is a Cell Wall Target in Aspergillus fumigatus

Publication Date:
23 Feb 2015

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Application of a novel regulatable Cre recombinase system to define the role of liver and gut metabolism in drug oral bioavailability.

Publication Date:
01 Feb 2015

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Dec 2014

Identification of Small Molecule Inhibitors of Pre-mRNA slicing

Publication Date:
12 Dec 2014

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Nov 2014

Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma brucei N-Myristoyltransferase Inhibitors: Identification and Evaluation of CNS Penetrant Compounds as Potential Treatments for Stage 2 Human African Trypanosomiasis

Publication Date:
20 Nov 2014

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Application of a novel regulatable Cre recombinase system to define the role of liver and gut metabolism in drug oral bioavailability.

Publication Date:
07 Nov 2014

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Respiratory Flexibility in Response to Inhibition of Cytochrome c Oxidase in Mycobacterium tuberculosis

Publication Date:
03 Nov 2014

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Sep 2014

The Design and Synthesis of Potent and Selective Inhibitors of Trypanosoma brucei Glycogen Synthase Kinase 3 for the Treatment of Human African Trypanosomiasis.

Publication Date:
08 Sep 2014

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A Target Repurposing Approach Identifies N-myristoyltransferase as a New Candidate Drug Target in Filarial Nematodes

Publication Date:
01 Sep 2014

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Jan 2014

Bisubstrate UDP–peptide conjugates as human O-GlcNAc transferase inhibitors

Publication Date:
26 Jan 2014

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Bisubstrate UDP–peptide conjugates as human O-GlcNAc transferase inhibitors

Publication Date:
26 Jan 2014

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Biochemical and genetic characterisation of Trypanosoma cruzi N-myristoyltransferase. Roberts AJ, Torrie LS, Wyllie S, Fairlamb AH.

Publication Date:
21 Jan 2014

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Biochemical and genetic characterisation of Trypanosoma cruzi N-myristoyltransferase.

Publication Date:
21 Jan 2014

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